99% Tianeptine soda iyọ CAS 30123-17-2
Sipesifikesonu
Nkan | ITOJU | Àbájáde |
Ifarahan | Funfun to yellowish lulú | Funfun okuta lulú |
Solubility | Tiotuka larọwọto Ninu omi ati kẹmika ati dichloromethane | Ni ibamu |
Idanimọ | Nipa IR, Lati baramu pẹlu boṣewa iṣẹ | Ni ibamu |
(2) O funni ni esi ti iṣuu soda | Ni ibamu | |
Awọn idoti A | ≤0.1% | Ko ri |
Awọn akojọpọ ti o jọmọ | Eyikeyi Max aimọ́ kan ṣoṣo≤0.1% | 0.060% |
Lapapọ awọn idoti≤0.4% | 0.36% | |
Awọn ojutu ti o ku (GC) | Acetidin≤ 0.5% | ND |
Dichloromethane≤ 0.06% | ND | |
Methanol≤ 0.3% | ND | |
Acetone ≤ 0.5% | 0.29% | |
Acetonitrile≤0.041% | 0.022% | |
Ethanol≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Omi | ≤ 5.0% | 3.8% |
Ayẹwo (HPLC) | 99.0% -101.0% (Lori anhydrousbasis) | 99.70% |
Ohun elo
Tianeptine iṣuu sodaiyọjẹ antidepressant tricyclic.Ilana antidepressant rẹ yatọ si ti awọn antidepressants tricyclic ibile.O le mu atunṣe ti 5-HT pọ si ni cleft synapti.Awọn ipa ti HT neuronal conduction.Ko si isunmọ fun choline tabi awọn olugba adrenergic.Ipa antidepressant jẹ iru si ti tricyclics, ṣugbọn ifarada dara ju ti awọn tricyclics lọ.Fun itọju ti irẹwẹsi, iwọntunwọnsi tabi ibanujẹ nla, neurogenic ati aibalẹ ifaseyin, aibalẹ ati aibanujẹ pẹlu ti ara, paapaa aibalẹ nipa ikun, ati aibalẹ ati aibalẹ ninu awọn alaisan ti o gbẹkẹle ọti-lile lakoko yiyọ kuro.